| Identification of pyrazolopyridazinones as PDEδ inhibitors B Papke, S Murarka, HA Vogel, P Martín-Gago, M Kovacevic, DC Truxius, ... Nature communications 7 (1), 11360, 2016 | 165 | 2016 |
| Stereoconvergent arylations and alkenylations of unactivated alkyl electrophiles: catalytic enantioselective synthesis of secondary sulfonamides and sulfones J Choi, P Martín-Gago, GC Fu Journal of the American Chemical Society 136 (34), 12161-12165, 2014 | 153 | 2014 |
| Arylfluorosulfate‐based electrophiles for covalent protein labeling: a new addition to the arsenal P Martín‐Gago, CA Olsen Angewandte Chemie International Edition 58 (4), 957-966, 2019 | 107 | 2019 |
| A PDE6δ‐KRas inhibitor chemotype with up to seven H‐bonds and picomolar affinity that prevents efficient inhibitor release by Arl2 P Martín‐Gago, EK Fansa, CH Klein, S Murarka, P Janning, M Schürmann, ... Angewandte Chemie 129 (9), 2463-2468, 2017 | 93 | 2017 |
| Covalent protein labeling at glutamic acids P Martín-Gago, EK Fansa, M Winzker, S Murarka, P Janning, ... Cell chemical biology 24 (5), 589-597. e5, 2017 | 81 | 2017 |
| MaxPHOS Ligand: PH/NH Tautomerism and Rhodium‐Catalyzed Asymmetric Hydrogenations E Cristobal‐Lecina, P Etayo, S Doran, M Reves, P Martín‐Gago, ... Advanced synthesis & catalysis 356 (4), 795-804, 2014 | 71 | 2014 |
| A tetradecapeptide somatostatin dicarba-analog: Synthesis, structural impact and biological activity P Martín-Gago, R Ramón, E Aragón, J Fernández-Carneado, ... Bioorganic & medicinal chemistry letters 24 (1), 103-107, 2014 | 35 | 2014 |
| Gas-phase collision induced dissociation mechanisms of peptides: Theoretical and experimental study of N-formylalanylamide fragmentation D Ortiz, P Martin-Gago, A Riera, K Song, JY Salpin, R Spezia International Journal of Mass Spectrometry 335, 33-44, 2013 | 35 | 2013 |
| Development of pyridazinone chemotypes targeting the PDEδ prenyl binding site S Murarka, P Martín‐Gago, C Schultz‐Fademrecht, A Al Saabi, ... Chemistry–A European Journal 23 (25), 6083-6093, 2017 | 29 | 2017 |
| Fine-tuning the [Pi]-[Pi]. Aromatic interactions in peptides: somatostatin analogues containing mesityl alanine P Martín-Gago, M Gomez-Caminals, R Ramón, X Verdaguer i Espaulella, ... Angewandte Chemie-International Edition, 2012, vol. 51, num. 8, p. 1820-1825, 2012 | 29 | 2012 |
| PDEδ inhibition impedes the proliferation and survival of human colorectal cancer cell lines harboring oncogenic KRas CH Klein, DC Truxius, HA Vogel, J Harizanova, S Murarka, ... International Journal of Cancer 144 (4), 767-776, 2019 | 28 | 2019 |
| Structure-based development of PDEδ inhibitors P Martín-Gago, EK Fansa, A Wittinghofer, H Waldmann Biological Chemistry 398 (5-6), 535-545, 2017 | 26 | 2017 |
| Insights into structure-activity relationships of somatostatin analogs containing mesitylalanine P Martín-Gago, E Aragón, M Gomez-Caminals, J Fernández-Carneado, ... Molecules 18 (12), 14564-14584, 2013 | 20 | 2013 |
| Aryl fluorosulfate based inhibitors that covalently target the SIRT5 lysine deacylase JE Bolding, P Martín‐Gago, N Rajabi, LF Gamon, TN Hansen, ... Angewandte Chemie International Edition 61 (47), e202204565, 2022 | 18 | 2022 |
| Arylfluorsulfat‐basierte Elektrophile für die kovalente Proteinmarkierung P Martín‐Gago, CA Olsen Angewandte Chemie 131 (4), 969-978, 2019 | 17 | 2019 |
| SSTR1‐and SSTR3‐Selective Somatostatin Analogues R Ramón, P Martín‐Gago, X Verdaguer, MJ Macias, P Martin‐Malpartida, ... ChemBioChem 12 (4), 625-632, 2011 | 16 | 2011 |
| Photo Cross‐Linking Probes Containing ϵ‐N‐Thioacyllysine and ϵ‐N‐Acyl‐(δ‐aza)lysine Residues M Bæk, P Martín‐Gago, JS Laursen, JLH Madsen, S Chakladar, CA Olsen Chemistry–A European Journal 26 (17), 3862-3869, 2020 | 14 | 2020 |
| Peptide aromatic interactions modulated by fluorinated residues: Synthesis, structure and biological activity of Somatostatin analogs containing 3-(3′, 5′ difluorophenyl)-alanine P Martín-Gago, Á Rol, T Todorovski, E Aragón, P Martin-Malpartida, ... Scientific Reports 6 (1), 27285, 2016 | 11 | 2016 |
| Nickel‐Electrocatalytic Decarboxylative Arylation to Access Quaternary Centers G Laudadio, P Neigenfind, Á Péter, CZ Rubel, MA Emmanuel, ... Angewandte Chemie International Edition 63 (8), e202314617, 2024 | 4 | 2024 |
| Ni-Electrocatalytic Decarboxylative Arylation to Access Quaternary Centers G Laudadio, P Neigenfind, Á Péter, CZ Rubel, MA Emmanuel, ... | 4 | 2023 |
