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Justina Kazokaitė-Adomaitienė
Justina Kazokaitė-Adomaitienė
The Netherlands Cancer Institute, Amsterdam
Verified email at nki.nl
Title
Cited by
Cited by
Year
Benzenesulfonamides with pyrimidine moiety as inhibitors of human carbonic anhydrases I, II, VI, VII, XII, and XIII
E Čapkauskaitė, A Zubrienė, A Smirnov, J Torresan, M Kišonaitė, ...
Bioorganic & medicinal chemistry 21 (22), 6937-6947, 2013
502013
Functionalization of fluorinated benzenesulfonamides and their inhibitory properties toward carbonic anhydrases
V Dudutienė, A Zubrienė, A Smirnov, DD Timm, J Smirnovienė, ...
ChemMedChem 10 (4), 662-687, 2015
432015
4-Amino-substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases
K Rutkauskas, A Zubrienė, I Tumosienė, K Kantminienė, M Kažemėkaitė, ...
Molecules 19 (11), 17356-17380, 2014
302014
Novel fluorinated carbonic anhydrase IX inhibitors reduce hypoxia-induced acidification and clonogenic survival of cancer cells
J Kazokaitė, R Niemans, V Dudutienė, HM Becker, J Leitāns, A Zubrienė, ...
Oncotarget 9 (42), 26800, 2018
252018
An update on anticancer drug development and delivery targeting carbonic anhydrase IX
J Kazokaitė, A Aspatwar, S Parkkila, D Matulis
PeerJ 5, e4068, 2017
252017
Intrinsic binding of 4‐substituted‐2, 3, 5, 6‐tetrafluorobenezenesulfonamides to native and recombinant human carbonic anhydrase VI
J Kazokaitė, G Milinavičiūtė, J Smirnovienė, J Matulienė, D Matulis
The FEBS Journal 282 (5), 972-983, 2015
222015
Fluorinated benzenesulfonamide anticancer inhibitors of carbonic anhydrase IX exhibit lower toxic effects on zebrafish embryonic development than ethoxzolamide
J Kazokaitė, A Aspatwar, V Kairys, S Parkkila, D Matulis
Drug and Chemical Toxicology 40 (3), 309-319, 2017
172017
Selective inhibition of human carbonic anhydrase IX in Xenopus oocytes and MDA-MB-231 breast cancer cells
J Kazokaitė, S Ames, HM Becker, JW Deitmer, D Matulis
Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup4), 38-44, 2016
122016
Actin maturation requires the ACTMAP/C19orf54 protease
P Haahr, RA Galli, LG van den Hengel, OB Bleijerveld, ...
Science 377 (6614), 1533-1537, 2022
102022
Engineered carbonic anhydrase VI-mimic enzyme switched the structure and affinities of inhibitors
J Kazokaitė, V Kairys, J Smirnovienė, A Smirnov, E Manakova, ...
Scientific reports 9 (1), 12710, 2019
42019
Engineering of chimeric carbonic anhydrases for designing isoform-selective inhibitors
J Smirnoviene, A Smirnov, V Kairys, J Kazokaite-Adomaitiene, ...
EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS 50 (SUPPL 1), 127-127, 2021
2021
Experimental approaches to identify selective picomolar inhibitors for carbonic anhydrase IX
J Kazokaitė-Adomaitienė, HM Becker, J Smirnovienė, LJ Dubois, ...
Current medicinal chemistry 28 (17), 3361-3384, 2021
2021
Development of fluorinated benzenesulfonamides as carbonic anhydrase IX inhibitors
V Dudutienė, A Zubrienė, J Kazokaitė, D Matulis
Chemistry and chemical technology: Lithuanian chemists conference, 2019 May …, 2019
2019
Efficacy of Novel CA IX Inhibitors in Biological Models
J Kazokaitė, HM Becker, HR Barker, A Aspatwar, S Parkkila, LJ Dubois, ...
Carbonic Anhydrase as Drug Target: Thermodynamics and Structure of Inhibitor …, 2019
2019
Investigation of human carbonic anhydrase VI and IX inhibitor efficacy and toxicity
J Kazokaitė
Vilniaus universitetas, 2018
2018
Discovery and Biological Characterization of Novel Selective Inhibitors of Carbonic Anhydrase IX
V Dudutienė, J Matulienė, A Smirnov, A Zubrienė, L Baranauskienė, ...
XIVth International conference of the Lithuanian biochemical society: the …, 2016
2016
Thermodynamics of anticancer drug lead binding to target proteins by thermal shift assay
A Zubrienė, J Gylytė, V Morkūnaitė, E Kazlauskas, L Baranauskienė, ...
Epigenetics–Bench to Bedside. COST Action TD0905: Program and Abstract Book …, 2013
2013
Thiophene sulfonamides as carbonic anhydrase inhibitors by titration calorimetry and thermal shift assay
V Morkūnaitė, A Zubrienė, L Baranauskienė, V Petrikaitė, J Gylytė, ...
Epigenetics: Bench to Bedside. COST Action TD0905: Abstract Book: April 26 …, 2012
2012
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