Benzenesulfonamides with pyrimidine moiety as inhibitors of human carbonic anhydrases I, II, VI, VII, XII, and XIII E Čapkauskaitė, A Zubrienė, A Smirnov, J Torresan, M Kišonaitė, ... Bioorganic & medicinal chemistry 21 (22), 6937-6947, 2013 | 53 | 2013 |
Functionalization of fluorinated benzenesulfonamides and their inhibitory properties toward carbonic anhydrases V Dudutienė, A Zubrienė, A Smirnov, DD Timm, J Smirnovienė, ... ChemMedChem 10 (4), 662-687, 2015 | 46 | 2015 |
4-Amino-substituted Benzenesulfonamides as Inhibitors of Human Carbonic Anhydrases K Rutkauskas, A Zubrienė, I Tumosienė, K Kantminienė, M Kažemėkaitė, ... Molecules 19 (11), 17356-17380, 2014 | 33 | 2014 |
Novel fluorinated carbonic anhydrase IX inhibitors reduce hypoxia-induced acidification and clonogenic survival of cancer cells J Kazokaitė, R Niemans, V Dudutienė, HM Becker, J Leitāns, A Zubrienė, ... Oncotarget 9 (42), 26800, 2018 | 32 | 2018 |
An update on anticancer drug development and delivery targeting carbonic anhydrase IX J Kazokaitė, A Aspatwar, S Parkkila, D Matulis PeerJ 5, e4068, 2017 | 26 | 2017 |
Intrinsic binding of 4‐substituted‐2, 3, 5, 6‐tetrafluorobenezenesulfonamides to native and recombinant human carbonic anhydrase VI J Kazokaitė, G Milinavičiūtė, J Smirnovienė, J Matulienė, D Matulis The FEBS Journal 282 (5), 972-983, 2015 | 25 | 2015 |
Fluorinated benzenesulfonamide anticancer inhibitors of carbonic anhydrase IX exhibit lower toxic effects on zebrafish embryonic development than ethoxzolamide J Kazokaitė, A Aspatwar, V Kairys, S Parkkila, D Matulis Drug and Chemical Toxicology 40 (3), 309-319, 2017 | 17 | 2017 |
Actin maturation requires the ACTMAP/C19orf54 protease P Haahr, RA Galli, LG van den Hengel, OB Bleijerveld, ... Science 377 (6614), 1533-1537, 2022 | 14 | 2022 |
Selective inhibition of human carbonic anhydrase IX in Xenopus oocytes and MDA-MB-231 breast cancer cells J Kazokaitė, S Ames, HM Becker, JW Deitmer, D Matulis Journal of Enzyme Inhibition and Medicinal Chemistry 31 (sup4), 38-44, 2016 | 12 | 2016 |
Engineered carbonic anhydrase VI-mimic enzyme switched the structure and affinities of inhibitors J Kazokaitė, V Kairys, J Smirnovienė, A Smirnov, E Manakova, ... Scientific reports 9 (1), 12710, 2019 | 10 | 2019 |
Picomolar fluorescent probes for compound affinity determination to carbonic anhydrase IX expressed in live cancer cells J Matulienė, G Žvinys, V Petrauskas, A Kvietkauskaitė, A Zakšauskas, ... Scientific reports 12 (1), 17644, 2022 | 7 | 2022 |
Identifying cross-lineage dependencies of cell-type specific regulators in gastruloids L Braccioli, T van den Brand, NA Saiz, C Fountas, PHN Celie, ... bioRxiv, 2022.11. 01.514697, 2022 | 2 | 2022 |
Experimental approaches to identify selective picomolar inhibitors for carbonic anhydrase IX J Kazokaitė-Adomaitienė, HM Becker, J Smirnovienė, LJ Dubois, ... Current medicinal chemistry 28 (17), 3361-3384, 2021 | 1 | 2021 |
JBP1 and JBP3 have conserved structures but different affinity to base-J I de Vries, A Adamopoulos, J Kazokaitė-Adomaitienė, T Heidebrecht, ... Journal of Structural Biology 217 (1), 108161, 2025 | | 2025 |
Protein Expression J Kazokaitė-Adomaitienė, PHN Celie Handbook of Molecular Biotechnology, 237-251, 2024 | | 2024 |
Engineering of chimeric carbonic anhydrases for designing isoform-selective inhibitors J Smirnoviene, A Smirnov, V Kairys, J Kazokaite-Adomaitiene, ... EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS 50 (SUPPL 1), 127-127, 2021 | | 2021 |
Development of fluorinated benzenesulfonamides as carbonic anhydrase IX inhibitors V Dudutienė, A Zubrienė, J Kazokaitė, D Matulis Chemistry and chemical technology: Lithuanian chemists conference, 2019 May …, 2019 | | 2019 |
Efficacy of Novel CA IX Inhibitors in Biological Models J Kazokaitė, HM Becker, HR Barker, A Aspatwar, S Parkkila, LJ Dubois, ... Carbonic Anhydrase as Drug Target: Thermodynamics and Structure of Inhibitor …, 2019 | | 2019 |
Investigation of human carbonic anhydrase VI and IX inhibitor efficacy and toxicity J Kazokaitė Vilniaus universitetas, 2018 | | 2018 |
Discovery and Biological Characterization of Novel Selective Inhibitors of Carbonic Anhydrase IX V Dudutienė, J Matulienė, A Smirnov, A Zubrienė, L Baranauskienė, ... XIVth International conference of the Lithuanian biochemical society: the …, 2016 | | 2016 |