Green, enzymatic syntheses of divanillin and diapocynin for the organic, biochemistry, or advanced general chemistry laboratory RT Nishimura, CH Giammanco, DA Vosburg Journal of Chemical Education 87 (5), 526-527, 2010 | 59 | 2010 |
Secondary alcohol quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,221,804, 2015 | 36 | 2015 |
Methylene linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,290,476, 2016 | 30 | 2016 |
Identification and structure activity relationships of quinoline tertiary alcohol modulators of RORγt DA Kummer, MD Cummings, M Abad, J Barbay, G Castro, R Wolin, ... Bioorganic & Medicinal Chemistry Letters 27 (9), 2047-2057, 2017 | 26 | 2017 |
Sustainable Practices in Medicinal Chemistry Part 2: Green by Design: Miniperspective I Aliagas, R Berger, K Goldberg, RT Nishimura, J Reilly, P Richardson, ... Journal of Medicinal Chemistry 60 (14), 5955-5968, 2017 | 25 | 2017 |
6-Substituted quinolines as RORγt inverse agonists JK Barbay, MD Cummings, M Abad, G Castro, KD Kreutter, DA Kummer, ... Bioorganic & Medicinal Chemistry Letters 27 (23), 5277-5283, 2017 | 24 | 2017 |
Phenyl linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,309,222, 2016 | 14 | 2016 |
Heteroaryl linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,303,015, 2016 | 11 | 2016 |
3-Substituted quinolines as RORγt inverse agonists VM Tanis, H Venkatesan, MD Cummings, M Albers, JK Barbay, K Herman, ... Bioorganic & Medicinal Chemistry Letters 29 (12), 1463-1470, 2019 | 10 | 2019 |
Quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,624,225, 2017 | 9 | 2017 |
Phenyl linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 10,369,146, 2019 | 7 | 2019 |
One-pot reductive alkylation of 2, 4-dihydroxy quinolines and pyridines PR Chheda, DA Kummer, RT Nishimura, KJ McClure, H Venkatesan The Journal of Organic Chemistry 86 (10), 7148-7162, 2021 | 6 | 2021 |
Methylene linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,284,308, 2016 | 6 | 2016 |
Phenyl and pyridinyl substituted imidazoles as modulators of RORγT S Goldberg, CL Martin, EG Fennema, DA Kummer, RT Nishimura, ... US Patent 11,345,666, 2022 | 5 | 2022 |
Phenyl linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,403,816, 2016 | 5 | 2016 |
HETEROARYL LINKED QUINOLINYL MODULATORS OF RORyt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent App. 14/053,707, 2014 | 5 | 2014 |
Phenyl substituted pyrazoles as modulators of RORγt S Goldberg, CL Martin, EG Fennema, DA Kummer, RT Nishimura, ... US Patent 10,975,037, 2021 | 4 | 2021 |
Heteroaryl linked quinolinyl modulators of RORgammat KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,328,095, 2016 | 4 | 2016 |
Alkyl linked quinolinyl modulators of RORγt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent 9,346,782, 2016 | 3 | 2016 |
HETEROARYL LINKED QUINOLINYL MODULATORS OF RORyt KA Leonard, K Barbay, JP Edwards, KD Kreutter, DA Kummer, ... US Patent App. 15/004,048, 2016 | 3 | 2016 |