| Antagonists of the P2X7 Receptor. From Lead Identification to Drug Development SD Guile, L Alcaraz, TN Birkinshaw, KC Bowers, MR Ebden, M Furber, ... Journal of medicinal chemistry 52 (10), 3123-3141, 2009 | 159 | 2009 |
| Class 1 PI3K clinical candidates and recent inhibitor design strategies: a medicinal chemistry perspective AE Garces, MJ Stocks Journal of medicinal chemistry 62 (10), 4815-4850, 2018 | 122 | 2018 |
| Molybdenum-mediated carbonylation of aryl halides with nucleophiles using microwave irradiation B Roberts, D Liptrot, L Alcaraz, T Luker, MJ Stocks Organic Letters 12 (19), 4280-4283, 2010 | 122 | 2010 |
| Pseudomonas aeruginosa Quorum Sensing Systems as Drug Discovery Targets: Current Position and Future Perspectives F Soukarieh, P Williams, MJ Stocks, M Camara Journal of medicinal chemistry 61 (23), 10385-10402, 2018 | 117 | 2018 |
| A synthesis of the C (1)-C (15) segment of tsukubaenolide (FK 506). P Kocienski, M Stocks, D Donald, M Cooper, A Manners Tetrahedron letters 29 (35), 4481-4484, 1988 | 103 | 1988 |
| Efficient and regiospecific one-pot synthesis of substituted 1, 2, 4-triazoles MJ Stocks, DR Cheshire, R Reynolds Organic Letters 6 (17), 2969-2971, 2004 | 99 | 2004 |
| Macrocyclic ring closures employing the intramolecular Heck reaction MJ Stocks, RP Harrison, SJ Teague Tetrahedron letters 36 (36), 6555-6558, 1995 | 90 | 1995 |
| In Silico and in Vitro-Guided Identification of Inhibitors of Alkylquinolone-Dependent Quorum Sensing in Pseudomonas aeruginosa F Soukarieh, E Vico Oton, JF Dubern, J Gomes, N Halliday, ... Molecules 23 (2), 257, 2018 | 61 | 2018 |
| Synthetic FKBP12 ligands. Design and synthesis of pyranose replacements. TN Birkenshaw, MV Caffrey, DE Cladingboel, ME Cooper, DK Donald, ... Bioorganic & Medicinal Chemistry Letters 4 (21), 2501-2506, 1994 | 60 | 1994 |
| Synthesis and evaluation of dual domain macrocyclic FKBP12 ligands. MV Caffrey, DE Cladingboel, ME Cooper, DK Donald, M Furber, ... Bioorganic & Medicinal Chemistry Letters 4 (21), 2507-2510, 1994 | 57 | 1994 |
| Modulators of CXCR4 and CXCR7/ACKR3 function I Adlere, B Caspar, M Arimont, S Dekkers, K Visser, J Stuijt, C de Graaf, ... Molecular pharmacology 96 (6), 737-752, 2019 | 54 | 2019 |
| Lipophilic activated ester prodrug approach for drug delivery to the intestinal lymphatic system JB Lee, A Zgair, J Malec, TH Kim, MG Kim, J Ali, C Qin, W Feng, M Chiang, ... Journal of controlled release 286, 10-19, 2018 | 54 | 2018 |
| The contribution to binding of the pyranoside substituents in the excised binding domain of FK-506 MJ Stocks, TN Birkinshaw, SJ Teague Bioorganic & Medicinal Chemistry Letters 4 (12), 1457-1460, 1994 | 52 | 1994 |
| The affinity of the excised binding domain of FK-506 for the immunophilin FKBP12. SJ Teague, MJ Stocks Bioorganic & Medicinal Chemistry Letters 3 (10), 1947-1950, 1993 | 51 | 1993 |
| The small molecule drug discovery process–from target selection to candidate selection M Stocks Introduction to biological and small molecule drug research and development …, 2013 | 50 | 2013 |
| Structure-driven HtL: design and synthesis of novel aminoindazole inhibitors of c-Jun N-terminal kinase activity MJ Stocks, S Barber, R Ford, F Leroux, S St-Gallay, S Teague, Y Xue Bioorganic & medicinal chemistry letters 15 (14), 3459-3462, 2005 | 50 | 2005 |
| The discovery of MMP7 inhibitors exploiting a novel selectivity trigger K Edman, M Furber, P Hemsley, C Johansson, G Pairaudeau, J Petersen, ... ChemMedChem 6 (5), 769-773, 2011 | 47 | 2011 |
| Molybdenum-mediated synthesis of quinazolin-4 (3H)-ones via cyclocarbonylation using microwave irradiation B Roberts, D Liptrot, T Luker, MJ Stocks, C Barber, N Webb, R Dods, ... Tetrahedron letters 52 (29), 3793-3796, 2011 | 45 | 2011 |
| A Practical Method for Targeted Library Design Balancing Lead‐like Properties with Diversity MJ Stocks, GRH Wilden, G Pairaudeau, MWD Perry, J Steele, ... ChemMedChem: Chemistry Enabling Drug Discovery 4 (5), 800-808, 2009 | 45 | 2009 |
| Novel quinazolinone inhibitors of the Pseudomonas aeruginosa quorum sensing transcriptional regulator PqsR S Grossman, F Soukarieh, W Richardson, R Liu, A Mashabi, J Emsley, ... European Journal of Medicinal Chemistry 208, 112778, 2020 | 44 | 2020 |
