Pretargeting in nuclear imaging and radionuclide therapy: improving efficacy of theranostics and nanomedicines EJL Stéen, PE Edem, K Nørregaard, JT Jørgensen, V Shalgunov, A Kjaer, ... Biomaterials 179, 209-245, 2018 | 167 | 2018 |
Comprehensive study of the drug delivery properties of poly (L-lactide)-poly (ethylene glycol) nanoparticles in rats and tumor-bearing mice V Shalgunov, D Zaytseva-Zotova, A Zintchenko, T Levada, Y Shilov, ... Journal of Controlled Release 261, 31-42, 2017 | 69 | 2017 |
Trans-cyclooctene-functionalized PeptoBrushes with improved reaction kinetics of the tetrazine ligation for pretargeted nuclear imaging EJL Stéen, JT Jørgensen, K Johann, K Norregaard, B Sohr, D Svatunek, ... ACS nano, 2019 | 68 | 2019 |
Agonist high-and low-affinity states of dopamine D2 receptors: methods of detection and clinical implications JP van Wieringen, J Booij, V Shalgunov, P Elsinga, MC Michel Naunyn-Schmiedeberg's archives of pharmacology 386 (2), 135-154, 2013 | 45 | 2013 |
The chemogenetic receptor ligand clozapine N-oxide induces in vivo neuroreceptor occupancy and reduces striatal glutamate levels S Bærentzen, A Casado-Sainz, D Lange, V Shalgunov, IM Tejada, ... Frontiers in neuroscience 13, 187, 2019 | 41 | 2019 |
Hunting for the high‐affinity state of G‐protein‐coupled receptors with agonist tracers: Theoretical and practical considerations for positron emission tomography imaging V Shalgunov, A van Waarde, J Booij, MC Michel, RAJO Dierckx, ... Medicinal research reviews 39 (3), 1014-1052, 2019 | 25 | 2019 |
Improved radiosynthesis and preliminary in vivo evaluation of the 11C-labeled tetrazine [11C] AE-1 for pretargeted PET imaging EJL Stéen, JT Jørgensen, IN Petersen, K Nørregaard, S Lehel, ... Bioorganic & medicinal chemistry letters 29 (8), 986-990, 2019 | 22 | 2019 |
In Vivo Veritas – 18F-radiolabeled glycomimetics allow insights into the pharmacological fate of galectin-3 inhibitors K Bratteby, E Torkelsson, E Tampio L'Estrade, K Peterson, V Shalgunov, ... Journal of Medicinal Chemistry, 2019 | 21 | 2019 |
Synthesis and Characterization of a Novel Series of Agonist Compounds as Potential Radiopharmaceuticals for Imaging Dopamine D2/3 Receptors in Their High … JP van Wieringen, V Shalgunov, HM Janssen, PM Fransen, AGM Janssen, ... Journal of medicinal chemistry 57 (2), 391-410, 2014 | 18 | 2014 |
Synthesis, Radiolabeling, and in Vitro and in Vivo Evaluation of [18F]ENL30: A Potential PET Radiotracer for the 5-HT7 Receptor E Tampio L’Estrade, FG Edgar, M Xiong, V Shalgunov, SL Baerentzen, ... Acs Omega 4 (4), 7344-7353, 2019 | 11 | 2019 |
Development and Evaluation of Two Potential 5-HT7 Receptor PET Tracers: [18F]ENL09 and [18F]ENL10 E Tampio L’Estrade, M Xiong, V Shalgunov, FG Edgar, B Volk, ... ACS chemical neuroscience 10 (9), 3961-3968, 2019 | 9 | 2019 |
Synthesis and evaluation in rats of the dopamine D2/3 receptor agonist 18F-AMC20 as a potential radioligand for PET V Shalgunov, JP van Wieringen, HM Janssen, PM Fransen, R Dierckx, ... J Nucl Med 56 (1), 133-9, 2015 | 9 | 2015 |
Synthesis and evaluation in rats of homologous series of [18F]-labeled dopamine D2/3 receptor agonists based on the 2-aminomethylchroman scaffold as potential PET tracers V Shalgunov, JP van Wieringen, HM Janssen, PM Fransen, RAJO Dierckx, ... EJNMMI research 5 (1), 41, 2015 | 8 | 2015 |
Convenient Entry to 18F‐Labeled Amines through the Staudinger Reduction EJL Stéen, V Shalgunov, C Denk, H Mikula, A Kjær, JL Kristensen, ... European journal of organic chemistry 2019 (8), 1722-1725, 2019 | 7 | 2019 |
Radiosynthesis and preclinical evaluation of [11C]Cimbi‐701 – Towards the imaging of cerebral 5‐HT7 receptors. ET L'Estrade, V Shalgunov, FG Edgar, MG Strebl‐Bantillo, M Xiong, ... Journal of Labelled Compounds and Radiopharmaceuticals, 2019 | 6 | 2019 |
New approaches to the immunotherapy of Alzheimer’s disease with the synthetic fragments of α7 subunit of the acetylcholine receptor OM Vol’pina, TD Volkova, MA Titova, YG Gershovich, NI Medvinskaya, ... Russian Journal of Bioorganic Chemistry 34 (1), 43-48, 2008 | 6 | 2008 |
Antibodies to synthetic fragments of nucleophosmin for the specific detection of its monomeric and oligomeric forms VS Shalgunov, NV Lobanova, TI Bulycheva, NL Deineko, TD Volkova, ... Russian journal of bioorganic chemistry 35 (6), 720, 2009 | 5 | 2009 |
Development of 18F-labeled agonist radioligands for PET imaging of the high-affinity state of cerebral dopamine D2/3 receptors V Shalgunov | 1 | 2017 |
Evaluation of [18F] AMC-15,[18F] FPr-AMC-13 and [18F] FEt-AMC-13 as candidate dopamine D2/3-agonist radioligands for PET V Shalgunov, JP van Wieringen, J Sijbesma, R Dierckx, M Michel, ... Journal of Nuclear Medicine 54 (supplement 2), 1108-1108, 2013 | 1 | 2013 |
Synthesis And Preliminary Evaluation Of [18F] AMC-20 As Candidate Dopamine D2/3-Agonist Radioligand For PET V Shalgunov, J van Wieringen, JWA Sijbesma, R Dierckx, MC Michel, ... EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING 40, S343-S343, 2013 | | 2013 |