| The medicinal chemist's toolbox for late stage functionalization of drug-like molecules T Cernak, KD Dykstra, S Tyagarajan, P Vachal, SW Krska Chemical Society Reviews 45 (3), 546-576, 2016 | 1276 | 2016 |
| Late‐stage functionalization of biologically active heterocycles through photoredox catalysis DA DiRocco, K Dykstra, S Krska, P Vachal, DV Conway, M Tudge Angewandte Chemie International Edition 53 (19), 4802-4806, 2014 | 439 | 2014 |
| Cobalt precursors for high-throughput discovery of base metal asymmetric alkene hydrogenation catalysts MR Friedfeld, M Shevlin, JM Hoyt, SW Krska, MT Tudge, PJ Chirik Science 342 (6162), 1076-1080, 2013 | 342 | 2013 |
| Highly efficient asymmetric synthesis of sitagliptin KB Hansen, Y Hsiao, F Xu, N Rivera, A Clausen, M Kubryk, S Krska, ... Journal of the American Chemical Society 131 (25), 8798-8804, 2009 | 301 | 2009 |
| Highly efficient synthesis of β-amino acid derivatives via asymmetric hydrogenation of unprotected enamines Y Hsiao, NR Rivera, T Rosner, SW Krska, E Njolito, F Wang, Y Sun, ... Journal of the American Chemical Society 126 (32), 9918-9919, 2004 | 293 | 2004 |
| The evolution of chemical high-throughput experimentation to address challenging problems in pharmaceutical synthesis SW Krska, DA DiRocco, SD Dreher, M Shevlin Accounts of chemical research 50 (12), 2976-2985, 2017 | 221 | 2017 |
| High-throughput optimization of Ir-catalyzed C–H borylation: a tutorial for practical applications SM Preshlock, B Ghaffari, PE Maligres, SW Krska, RE Maleczka Jr, ... Journal of the American Chemical Society 135 (20), 7572-7582, 2013 | 219 | 2013 |
| Unlocking the potential of asymmetric hydrogenation at Merck CS Shultz, SW Krska Accounts of chemical research 40 (12), 1320-1326, 2007 | 193 | 2007 |
| A Traceless Directing Group for C H Borylation SM Preshlock, DL Plattner, PE Maligres, SW Krska, RE Maleczka Jr, ... Angewandte Chemie 125 (49), 13153-13157, 2013 | 186 | 2013 |
| Chemistry informer libraries: a chemoinformatics enabled approach to evaluate and advance synthetic methods PS Kutchukian, JF Dropinski, KD Dykstra, B Li, DA DiRocco, ... Chemical science 7 (4), 2604-2613, 2016 | 164 | 2016 |
| Zirconium-mediated metathesis of imines: A study of the scope, longevity, and mechanism of a complicated catalytic system RL Zuckerman, SW Krska, RG Bergman Journal of the American Chemical Society 122 (5), 751-761, 2000 | 150 | 2000 |
| Silyl phosphorus and nitrogen donor chelates for homogeneous ortho borylation catalysis B Ghaffari, SM Preshlock, DL Plattner, RJ Staples, PE Maligres, SW Krska, ... Journal of the American Chemical Society 136 (41), 14345-14348, 2014 | 148 | 2014 |
| Synthesis of water-soluble carbosilane dendrimers SW Krska, D Seyferth Journal of the American Chemical Society 120 (15), 3604-3612, 1998 | 126 | 1998 |
| Reaction development and mechanistic study of a ruthenium catalyzed intramolecular asymmetric reductive amination en route to the dual orexin inhibitor Suvorexant (MK-4305) NA Strotman, CA Baxter, KMJ Brands, E Cleator, SW Krska, RA Reamer, ... Journal of the American Chemical Society 133 (21), 8362-8371, 2011 | 119 | 2011 |
| Designed Ligands as Probes for the Catalytic Binding Mode in Mo‐Catalyzed Asymmetric Allylic Alkylation BM Trost, K Dogra, I Hachiya, T Emura, DL Hughes, S Krska, RA Reamer, ... Angewandte Chemie 114 (11), 2009-2012, 2002 | 118 | 2002 |
| Photoredox-catalyzed hydroxymethylation of heteroaromatic bases CA Huff, RD Cohen, KD Dykstra, E Streckfuss, DA DiRocco, SW Krska The Journal of Organic Chemistry 81 (16), 6980-6987, 2016 | 114 | 2016 |
| Pharmaceutical diversification via palladium oxidative addition complexes MR Uehling, RP King, SW Krska, T Cernak, SL Buchwald Science 363 (6425), 405-408, 2019 | 111 | 2019 |
| Reversed-polarity synthesis of diaryl ketones via palladium-catalyzed cross-coupling of acylsilanes JR Schmink, SW Krska Journal of the American Chemical Society 133 (49), 19574-19577, 2011 | 105 | 2011 |
| C (sp3)–H methylation enabled by peroxide photosensitization and Ni-mediated radical coupling A Vasilopoulos, SW Krska, SS Stahl Science 372 (6540), 398-403, 2021 | 103 | 2021 |
| Copper-catalysed benzylic C–H coupling with alcohols via radical relay enabled by redox buffering H Hu, SJ Chen, M Mandal, SM Pratik, JA Buss, SW Krska, CJ Cramer, ... Nature catalysis 3 (4), 358-367, 2020 | 100 | 2020 |
Edward GrabowskiMerck Research Labs, Vice President of Chemistry RetiredVerified email at alum.mit.edu
