Shane W. Krska
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The medicinal chemist's toolbox for late stage functionalization of drug-like molecules
T Cernak, KD Dykstra, S Tyagarajan, P Vachal, SW Krska
Chemical Society Reviews 45 (3), 546-576, 2016
Late‐stage functionalization of biologically active heterocycles through photoredox catalysis
DA DiRocco, K Dykstra, S Krska, P Vachal, DV Conway, M Tudge
Angewandte Chemie International Edition 53 (19), 4802-4806, 2014
Cobalt precursors for high-throughput discovery of base metal asymmetric alkene hydrogenation catalysts
MR Friedfeld, M Shevlin, JM Hoyt, SW Krska, MT Tudge, PJ Chirik
Science 342 (6162), 1076-1080, 2013
Highly efficient asymmetric synthesis of sitagliptin
KB Hansen, Y Hsiao, F Xu, N Rivera, A Clausen, M Kubryk, S Krska, ...
Journal of the American Chemical Society 131 (25), 8798-8804, 2009
Highly efficient synthesis of β-amino acid derivatives via asymmetric hydrogenation of unprotected enamines
Y Hsiao, NR Rivera, T Rosner, SW Krska, E Njolito, F Wang, Y Sun, ...
Journal of the American Chemical Society 126 (32), 9918-9919, 2004
The evolution of chemical high-throughput experimentation to address challenging problems in pharmaceutical synthesis
SW Krska, DA DiRocco, SD Dreher, M Shevlin
Accounts of chemical research 50 (12), 2976-2985, 2017
High-throughput optimization of Ir-catalyzed C–H borylation: a tutorial for practical applications
SM Preshlock, B Ghaffari, PE Maligres, SW Krska, RE Maleczka Jr, ...
Journal of the American Chemical Society 135 (20), 7572-7582, 2013
Unlocking the potential of asymmetric hydrogenation at Merck
CS Shultz, SW Krska
Accounts of chemical research 40 (12), 1320-1326, 2007
A Traceless Directing Group for C H Borylation
SM Preshlock, DL Plattner, PE Maligres, SW Krska, RE Maleczka Jr, ...
Angewandte Chemie 125 (49), 13153-13157, 2013
Chemistry informer libraries: a chemoinformatics enabled approach to evaluate and advance synthetic methods
PS Kutchukian, JF Dropinski, KD Dykstra, B Li, DA DiRocco, ...
Chemical science 7 (4), 2604-2613, 2016
Zirconium-mediated metathesis of imines: A study of the scope, longevity, and mechanism of a complicated catalytic system
RL Zuckerman, SW Krska, RG Bergman
Journal of the American Chemical Society 122 (5), 751-761, 2000
Silyl phosphorus and nitrogen donor chelates for homogeneous ortho borylation catalysis
B Ghaffari, SM Preshlock, DL Plattner, RJ Staples, PE Maligres, SW Krska, ...
Journal of the American Chemical Society 136 (41), 14345-14348, 2014
Synthesis of water-soluble carbosilane dendrimers
SW Krska, D Seyferth
Journal of the American Chemical Society 120 (15), 3604-3612, 1998
Reaction development and mechanistic study of a ruthenium catalyzed intramolecular asymmetric reductive amination en route to the dual orexin inhibitor Suvorexant (MK-4305)
NA Strotman, CA Baxter, KMJ Brands, E Cleator, SW Krska, RA Reamer, ...
Journal of the American Chemical Society 133 (21), 8362-8371, 2011
Designed Ligands as Probes for the Catalytic Binding Mode in Mo‐Catalyzed Asymmetric Allylic Alkylation
BM Trost, K Dogra, I Hachiya, T Emura, DL Hughes, S Krska, RA Reamer, ...
Angewandte Chemie 114 (11), 2009-2012, 2002
Photoredox-catalyzed hydroxymethylation of heteroaromatic bases
CA Huff, RD Cohen, KD Dykstra, E Streckfuss, DA DiRocco, SW Krska
The Journal of Organic Chemistry 81 (16), 6980-6987, 2016
Pharmaceutical diversification via palladium oxidative addition complexes
MR Uehling, RP King, SW Krska, T Cernak, SL Buchwald
Science 363 (6425), 405-408, 2019
Reversed-polarity synthesis of diaryl ketones via palladium-catalyzed cross-coupling of acylsilanes
JR Schmink, SW Krska
Journal of the American Chemical Society 133 (49), 19574-19577, 2011
C (sp3)–H methylation enabled by peroxide photosensitization and Ni-mediated radical coupling
A Vasilopoulos, SW Krska, SS Stahl
Science 372 (6540), 398-403, 2021
Copper-catalysed benzylic C–H coupling with alcohols via radical relay enabled by redox buffering
H Hu, SJ Chen, M Mandal, SM Pratik, JA Buss, SW Krska, CJ Cramer, ...
Nature catalysis 3 (4), 358-367, 2020
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